Oxametacin

Oxametacin

SCHEMBL24552

COc1ccc2c(c1)c(CC(=O)NO)c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 1.00
PTGS2 P35354 12/20 0.85
AKR1C3 P42330 3/20 0.81
CNR2 P34972 1/20 0.81
MAPT P10636 3/20 0.80
KMT2A Q03164 2/20 0.80
NPSR1 Q6W5P4 2/20 0.80
AKR1C2 P52895 2/20 0.79
KDM4E B2RXH2 1/20 0.79
MEN1 O00255 1/20 0.79
PTGES O14684 1/20 0.79
ABCC3 O15438 1/20 0.79
ABCC4 O15439 1/20 0.79
ABCB11 O95342 1/20 0.79
MT-CO2 P00403 1/20 0.79
LMNA P02545 1/20 0.79
ALB P02768 1/20 0.79
CYP1A2 P05177 1/20 0.79
ABCB1 P08183 1/20 0.79
ALOX5 P09917 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxametacin SCHEMBL29378857 1.00 PTGS1 (1.00) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL14405006 0.92 PTGS2 (1.00) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL20259394 0.91 PTGS2 (0.83) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL9657228 0.91 PTGS1 (0.85) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL14398315 0.90 PTGS1 (0.82) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL5107049 0.90 PTGS2 (0.82) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL5112013 0.90 PTGS2 (0.84) PTGS1PTGS2
SCHEMBL30426824 0.89 PTGS2 (1.00) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL14086813 0.89 PTGS2 (1.00) PTGS1PTGS2AKR1C3CNR2MAPT
SCHEMBL17378074 0.89 PTGS2 (0.80) PTGS1PTGS2AKR1C3CNR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1944 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
EP-2709663-B1 USE OF ANTI-CGRP ANTIBODIES AND ANTIBODY FRAGMENTS TO PREVENT OR INHIBIT PHOTOPHOBIA OR LIGHT AVERSION IN SUBJECTS IN NEED THEREOF, ESPECIALLY MIGRAINE SUFFERERS ALDERBIO HOLDINGS LLC (US) 2019-03-20 EP claimed
US-20170128383-A1 Polymeric Adhesive Matrix with Salified Carboxylic Groups for Transdermal Use BOUTY S.P.A. (IT) 2017-05-11 US claimed
CN-102292106-B IL-6 antibody and uses thereof ALDER BIOPHARMACEUTICALS, INC. (US) 2016-02-03 CN claimed
US-8865198-B2 Method for treating a periodontal disease DEXCEL PHARMA TECHNOLOGIES LTD. (IL) 2014-10-21 US claimed
US-20140080911-A1 Polymeric Adhesive Matrix with Salified Carboxylic Groups for Transdermal Use BOUTY S P A (IT) 2014-03-20 US claimed
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP claimed
US-8361492-B2 Drug delivery system and methods of use Ocugenics, LLC (US) 2013-01-29 US claimed
EP-2455064-A1 Device for treating a periodontal disease Dexcel Pharma Technologies Ltd. (IL) 2012-05-23 EP claimed
EP-2448558-A1 LOCAL THERAPEUTIC RELEASE DEVICE Dexcel Pharma Technologies Ltd. (IL) 2012-05-09 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP claimed
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
US-4455432-A Process for the preparation of 1-(4-chloro-benzoyl)-5-methoxy-2-methyl-3-indolyl-acetohydroxamic acid UNIBIOS S.P.A. (IT) 1984-06-19 US claimed