SCHEMBL245783

SCHEMBL245783

NCc1ncco1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL243025 0.97
Hydrochloric Acid SCHEMBL20532707 0.97
Trifluoroacetic Acid SCHEMBL27610628 0.82 L3MBTL1 (0.36)
SCHEMBL659550 0.80
Hydrochloric Acid SCHEMBL14743990 0.78 HRH1 (0.34)
Hydrochloric Acid SCHEMBL26111974 0.78
SCHEMBL29086344 0.78 CYP1B1 (0.32)
SCHEMBL7704422 0.78 CYP1B1 (0.32)
SCHEMBL11005395 0.77
SCHEMBL8569658 0.75 HRH1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 418 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114213395-B Pyrimidone acyl piperazine compound and preparation method and application thereof 山东大学 2022-10-25 CN claimed
CN-110698420-B Preparation method of 2-oxazole methylamine heterocyclic compound 上海阿拉丁生化科技股份有限公司 2022-10-14 CN claimed
CN-114213395-A Pyrimidone acyl piperazine compound and preparation method and application thereof 山东大学 2022-03-22 CN claimed
CN-110698420-A Preparation method of 2-oxazole methylamine heterocyclic compound 上海阿拉丁生化科技股份有限公司 2020-01-17 CN claimed
EP-3510404-A1 CHEMICAL PROBES OF LYSYL OXIDASE-LIKE 2 AND USES THEREOF Pharmakea, Inc. (US) 2019-07-17 EP claimed
US-20190192697-A1 CHEMICAL PROBES OF LYSYL OXIDASK-LIKE 2 AND USES THEREOF PHARMAKEA, INC. 2019-06-27 US claimed
CN-109574948-A A kind of preparation method of bis- (tertbutyloxycarbonyl) amine 凯瑞斯德生化(苏州)有限公司 2019-04-05 CN claimed
CN-108884049-A 2 inhibitor of quinolinone lysyloxidase sample and application thereof 法玛克亚公司 2018-11-23 CN claimed
WO-2018048928-A1 CHEMICAL PROBES OF LYSYL OXIDASE-LIKE 2 AND USES THEREOF PHARMAKEA, INC. (US) 2018-03-15 WO claimed
US-20140235548-A1 COMPOSITIONS AND METHODS FOR JAMM PROTEIN INHIBITION CLEAVE BIOSCIENCES, INC. (US) 2014-08-21 US claimed
US-7462604-B2 Hair growth promotor composition LION CORPORATION (JP) 2008-12-09 US claimed
US-20080207683-A1 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. 2008-08-28 US claimed
WO-2008100622-A2 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. (US) 2008-08-21 WO claimed
US-20080182870-A1 PYRIDO(3,2-d)PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-07-31 US claimed
WO-2008077651-A1 PYRIDO(3,2-D)PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-07-03 WO claimed
WO-2008020024-A1 NTETRAHYDROPYRIDOTHIOPHENE DERIVATIVES FOR THE TREATMENT OF CANCER 4SC AG (DE) 2008-02-21 WO claimed
US-20070116657-A1 Hair growth promotor composition LION CORPORATION (JP) 2007-05-24 US claimed
EP-1671616-A1 HAIR TONIC COMPOSITION Lion Corporation (JP) 2006-06-21 EP claimed
EP-0540854-B1 Preparation for promoting hair growth SANSHO SEIYAKU KK (JP) 1998-01-21 EP claimed
EP-0540854-A2 Preparation for promoting hair growth Sansho Seiyaku Co., Ltd. (JP) 1993-05-12 EP claimed