SCHEMBL24596309

SCHEMBL24596309

O=c1c2[nH]ncc2c2ccc(C(F)(F)F)nc2n1-c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 16/20 0.58
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
METAP2 P50579 2/20 0.38
S1PR4 O95977 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
S1PR1 P21453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30649344 1.00 MAT2A (0.58) MAT2AKDM4EALDH1A1METAP2S1PR4
SCHEMBL24596312 0.91 MAT2A (0.58) MAT2AKDM4EALDH1A1METAP2
SCHEMBL24596220 0.83 MAT2A (0.59) MAT2AKDM4EALDH1A1S1PR4GLA
SCHEMBL24596241 0.82 MAT2A (0.60) MAT2AKDM4EALDH1A1S1PR4GLA
SCHEMBL24596273 0.78 MAT2A (0.58) MAT2AKDM4EALDH1A1S1PR4GLA
SCHEMBL24596307 0.78 MAT2A (0.58) MAT2A
SCHEMBL27295076 0.78 MAT2A (0.78) MAT2A
SCHEMBL24596200 0.77 MAT2A (0.57) MAT2AALDH1A1
SCHEMBL24596196 0.77 MAT2A (0.57) MAT2AALDH1A1
SCHEMBL28874822 0.77 MAT2A (0.59) MAT2AKDM4EALDH1A1S1PR4GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240124454-A1 TRICYCLIC COMPOUND AND USE THEREOF NANJING ZAIMING PHARMACEUTICAL CO., LTD. (CN) 2024-04-18 US disclosed
EP-4273146-A1 TRICYCLIC COMPOUND AND USE THEREOF Nanjing Zaiming Pharmaceutical Co., Ltd. (CN) 2023-11-08 EP disclosed
EP-4273146-A1 TRICYCLIC COMPOUND AND USE THEREOF Nanjing Zaiming Pharmaceutical Co., Ltd. (CN) 2023-11-08 EP disclosed
WO-2022143864-A1 TRICYCLIC COMPOUND AND USE THEREOF 江苏先声药业有限公司 2022-07-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124454-A1 TRICYCLIC COMPOUND AND USE THEREOF MAT2A, MNAT1, KAT2A MAT2A 1/4885KDM4E 2337/4885ALDH1A1 1518/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.