SCHEMBL24601143

SCHEMBL24601143

C/C=C\c1ccncc1/C=C/C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
APLNR P35414 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
HMGCR P04035 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTT P42858 1/20 0.31
CYP1A1 P04798 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24248359 1.00 CCNC (0.35) CCNCCDK8APLNRCYP11B1CYP11B2
SCHEMBL12508937 0.87 IMPDH2 (0.33) CCNCCDK8
SCHEMBL18381481 0.87 IMPDH2 (0.36) CCNCCDK8HTT
SCHEMBL26750323 0.84 CCNC (0.30) CCNCCDK8
SCHEMBL14822507 0.82 TRPA1 (0.35) CCNCCDK8APLNRCYP11B1CYP11B2
SCHEMBL21881933 0.82 TRPA1 (0.35) CCNCCDK8APLNRCYP11B1CYP11B2
SCHEMBL14822558 0.82 SIRT3 (0.38) APLNRCYP11B1CYP11B2CYP3A4
SCHEMBL20691108 0.81 CHRNB2 (0.32)
SCHEMBL18716205 0.80 GAA (0.43) CCNCCDK8CYP11B1CYP11B2CYP3A4
SCHEMBL16130317 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4273153-A1 ADENOSINE A3 RECEPTOR AGONISTS, PREPARATION METHODS AND USES THEREOF Zhejiang Vimgreen Pharmaceuticals, Ltd (CN) 2023-11-08 EP disclosed
WO-2022143740-A1 ADENOSINE A3 RECEPTOR AGONIST, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江春禾医药科技有限公司 2022-07-07 WO disclosed