SCHEMBL24616474

SCHEMBL24616474

CC(C)c1cccn2cc(N)nc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.35
HSD11B1 P28845 1/20 0.35
NPC1 O15118 6/20 0.35
RAB9A P51151 6/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
KDM4E B2RXH2 3/20 0.35
TP53 P04637 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HSD17B10 Q99714 2/20 0.35
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
DHFR P00374 1/20 0.33
PKM P14618 1/20 0.33
ALDH1A2 O94788 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24371127 0.81 HTR4 (0.42) NR1I2HSD11B1NPC1RAB9AALDH1A1
SCHEMBL27017623 0.80 HTR4 (0.35) NR1I2HSD11B1NPC1RAB9AALDH1A1
SCHEMBL21348795 0.77 SMN1; SMN2 (0.40) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL24615934 0.72 NPC1 (0.35) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL26701981 0.69 NPC1 (0.46) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL2605414 0.69 NUDT1 (0.41) NR1I2HSD11B1HPGDTSHRPIK3CG
SCHEMBL11031081 0.69 USP7 (0.43) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL21348767 0.68 ALDH1A1 (0.47) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL6269053 0.68 NR1I2 (0.40) NR1I2HSD11B1KDM4EHSD17B10HPGD
SCHEMBL24368132 0.68 ALDH1A1 (0.46) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022148422-A1 BRIDGED COMPOUNDS AS KRAS G12D INHIBITOR AND DEGRADER AND THE USE THEREOF BEIGENE, LTD. (KY) 2022-07-14 WO disclosed