SCHEMBL24620331

SCHEMBL24620331

NC(=O)CCC(N)(O)C(=O)N1CCC2(CCNC2=O)CC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OTUD7B Q6GQQ9 1/20 0.35
IDO1 P14902 1/20 0.34
CALCRL Q16602 1/20 0.32
CDK8 P49336 6/20 0.32
CCNC P24863 5/20 0.32
SPR P35270 1/20 0.31
CDK19 Q9BWU1 1/20 0.30
PIK3CA P42336 1/20 0.30
MTOR P42345 1/20 0.30
KCNH2 Q12809 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24620526 0.86 OTUD7B (0.35) OTUD7BCALCRLCDK8CCNCSPR
SCHEMBL19852883 0.78 ITGB3 (0.42) OTUD7BCALCRL
SCHEMBL29890275 0.75 OTUD7B (0.46) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL18702126 0.74 OTUD7B (0.43) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL24338486 0.73 OTUD7B (0.36) OTUD7BCALCRLCDK8CCNCSPR
SCHEMBL19852880 0.71 OTUD7B (0.43) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL19852881 0.71 OTUD7B (0.43) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL4072997 0.70 OTUD7B (0.47) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL19852884 0.69 OTUD7B (0.39) OTUD7BIDO1CALCRLCDK8CCNC
SCHEMBL18711886 0.69 OTUD7B (0.46) OTUD7BCDK8CCNCSPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312591-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF TENACIA BIOTECHNOLOGY (HONG KONG) CO., LIMITED (HK) 2023-10-05 US disclosed
US-11530223-B2 Spiro-lactam NMDA receptor modulators and uses thereof APTINYX INC. (US) 2022-12-20 US disclosed
US-20220220119-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF TENACIA BIOTECHNOLOGY (HONG KONG) CO., LIMITED (HK) 2022-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11530223-B2 Spiro-lactam NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885IDO1 2875/4885CALCRL 981/4885
US-20220220119-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885IDO1 2875/4885CALCRL 981/4885
US-20230312591-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885IDO1 2875/4885CALCRL 981/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.