SCHEMBL24620526

SCHEMBL24620526

C[C@@](N)(CCC(N)=O)C(=O)N1CCC2(CCNC2=O)CC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OTUD7B Q6GQQ9 1/20 0.35
CDK8 P49336 10/20 0.33
CCNC P24863 9/20 0.33
SPR P35270 1/20 0.32
CDK19 Q9BWU1 2/20 0.32
CALCRL Q16602 1/20 0.32
TYK2 P29597 3/20 0.31
JAK1 P23458 2/20 0.31
JAK2 O60674 1/20 0.30
JAK3 P52333 1/20 0.30
SLC34A1 Q06495 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24620331 0.86 OTUD7B (0.35) OTUD7BCDK8CCNCSPRCDK19
SCHEMBL18702126 0.79 OTUD7B (0.43) OTUD7BCDK8CCNCSPRCALCRL
SCHEMBL19852883 0.77 ITGB3 (0.42) OTUD7BCALCRL
SCHEMBL19852926 0.76 GRIN2B (0.31)
SCHEMBL29890275 0.74 OTUD7B (0.46) OTUD7BCDK8CCNCSPRCALCRL
SCHEMBL24338486 0.72 OTUD7B (0.36) OTUD7BCDK8CCNCSPRCALCRL
SCHEMBL745671 0.72 OTUD7B (0.40) OTUD7BCDK8CCNCSPRCDK19
SCHEMBL19852884 0.71 OTUD7B (0.39) OTUD7BCDK8CCNCSPRCDK19
SCHEMBL18711886 0.71 OTUD7B (0.46) OTUD7BCDK8CCNCSPRTYK2
SCHEMBL19852881 0.70 OTUD7B (0.43) OTUD7BCDK8CCNCSPRCALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312591-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF TENACIA BIOTECHNOLOGY (HONG KONG) CO., LIMITED (HK) 2023-10-05 US disclosed
US-11530223-B2 Spiro-lactam NMDA receptor modulators and uses thereof APTINYX INC. (US) 2022-12-20 US disclosed
US-20220220119-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF TENACIA BIOTECHNOLOGY (HONG KONG) CO., LIMITED (HK) 2022-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11530223-B2 Spiro-lactam NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885CDK8 1003/4885CCNC 2764/4885
US-20220220119-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885CDK8 1003/4885CCNC 2764/4885
US-20230312591-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN3A OTUD7B 3931/4885CDK8 1003/4885CCNC 2764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.