SCHEMBL24625565

SCHEMBL24625565

COC(=O)c1ccc(OC)c(-c2ccc(O)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.58
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA7 P43166 2/20 0.58
CA9 Q16790 2/20 0.58
CA14 Q9ULX7 2/20 0.58
MAPT P10636 5/20 0.54
HPSE Q9Y251 1/20 0.49
KMT2A Q03164 3/20 0.49
EGFR P00533 1/20 0.49
XDH P47989 1/20 0.49
ERN1 O75460 1/20 0.48
PTGS2 P35354 1/20 0.47
GAA P10253 2/20 0.46
MGAM O43451 1/20 0.46
SI P14410 1/20 0.46
MGAM2 Q2M2H8 1/20 0.46
MEN1 O00255 2/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6248649 0.86 LMNA (0.59) CA12CA1CA2CA7CA9
SCHEMBL35823 0.86 PTGS2 (0.58) MAPTKMT2AEGFRPTGS2MEN1
SCHEMBL3631102 0.85 CA1 (0.51) CA12CA1CA2CA7CA9
SCHEMBL6702060 0.85 CA1 (0.63) CA12CA1CA2CA7CA9
SCHEMBL13276414 0.82 AR (0.57) MAPTKMT2AERN1PTGS2RAB9A
SCHEMBL3631211 0.81 LMNA (0.56) MAPTEGFRPTGS2GAAMGAM
SCHEMBL6704931 0.80 PTGS1 (0.55) MAPTKMT2AERN1MEN1RAB9A
SCHEMBL6883774 0.79 HSD17B1 (0.59) CA12CA1CA2CA7CA9
SCHEMBL17559286 0.79 ABL1 (0.61) MAPTKMT2AEGFRERN1
SCHEMBL7501527 0.79 EGFR (0.69) MAPTKMT2AEGFRERN1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022149925-A1 NOVEL TRYPTOPHAN HYDROXYLASE INHIBITOR AND USE THEREOF 광주과학기술원 2022-07-14 WO disclosed
WO-2022149925-A1 NOVEL TRYPTOPHAN HYDROXYLASE INHIBITOR AND USE THEREOF 광주과학기술원 2022-07-14 WO disclosed