SCHEMBL24629934

SCHEMBL24629934

CN(C)CCOc1ccc(NC(=O)CN(C)C(=O)OC(C)(C)C)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.53
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
CHRM1 P11229 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
DRD1 P21728 1/20 0.46
HRH2 P25021 1/20 0.46
HTR1B P28222 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HRH1 P35367 1/20 0.46
DRD3 P35462 1/20 0.46
MCHR2 Q969V1 1/20 0.46
MCHR1 Q99705 1/20 0.46
MAOA P21397 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29769200 1.00 KDR (0.53) KDRCHRM2ADRA2ACHRM1ADRA2B
SCHEMBL29769183 0.86 ALDH1A1 (0.58) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL24629451 0.86 ALDH1A1 (0.58) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL24629958 0.79 KDR (0.57) KDRCHRM2ADRA2ACHRM1ADRA2B
SCHEMBL29769152 0.79 KDR (0.57) KDRCHRM2ADRA2ACHRM1ADRA2B
SCHEMBL7499427 0.77 ALDH1A1 (0.56) MCHR1ALDH1A1MEN1KMT2AHTT
SCHEMBL24630015 0.77 LMNA (0.46) MCHR1ALDH1A1KDM4EGAAMEN1
SCHEMBL21601484 0.76 MAPK1 (0.51) MAOAALDH1A1KDM4EGAAMAPK1
SCHEMBL21601488 0.75 KDM4E (0.55) CHRM1ALDH1A1KDM4EGAAMAPK1
SCHEMBL4015052 0.74 PDK2 (0.43) CHRM2HTR2CMAOAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022150574-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2022-07-14 WO disclosed