SCHEMBL24630261

SCHEMBL24630261

N#Cc1cc2cccc(Br)c2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
DYRK1A Q13627 4/20 0.42
NOS1 P29475 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
NUDT1 P36639 1/20 0.33
CLK1 P49759 1/20 0.32
DAO P14920 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
MAP2K2 P36507 1/20 0.30
MAP2K1 Q02750 1/20 0.30
CDK9 P50750 1/20 0.30
DYRK2 Q92630 1/20 0.30
DYRK1B Q9Y463 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28726348 0.79 DAO (0.50) CA12CA9DYRK1ANOS1HRH4
SCHEMBL20504985 0.78 DAO (0.49) CA12CA9DYRK1AHRH4NUDT1
SCHEMBL28907064 0.74 ALDH1A1 (0.49) DYRK1ACLK1KDM4EALDH1A1HPGD
SCHEMBL21877855 0.74 CA12 (0.53) CA12CA9DYRK1ANOS1HRH4
SCHEMBL24629881 0.73 XDH (0.46) ALDH1A1MAPT
SCHEMBL29769118 0.73 XDH (0.46) ALDH1A1MAPT
SCHEMBL17673224 0.72 CA12 (0.52) CA12CA9DYRK1ANOS1HRH4
SCHEMBL6505957 0.71 CA12 (0.50) CA12CA9DYRK1ANOS1HRH4
SCHEMBL597517 0.71 CA12 (0.50) CA12CA9DYRK1ANOS1HRH4
SCHEMBL993313 0.70 AHR (0.41) DYRK1ANOS1HRH4NUDT1CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022150574-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2022-07-14 WO disclosed