SCHEMBL2463548

SCHEMBL2463548

BrN1CCN(c2ccc3ncc4nncn4c3c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.36
TP53 P04637 5/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
HRH4 Q9H3N8 2/20 0.34
HRH3 Q9Y5N1 2/20 0.34
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
POLB P06746 2/20 0.33
LCK P06239 4/20 0.33
C1S P09871 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL439463 0.99 MAPT (0.35) MAPTTP53SMN1; SMN2KMT2AMEN1
SCHEMBL29821277 0.68 HSD17B10 (0.49) MAPTSMN1; SMN2KMT2AGLAGAA
SCHEMBL1602168 0.68 HSD17B10 (0.49) MAPTSMN1; SMN2KMT2AGLAGAA
SCHEMBL21642536 0.65 SMN1; SMN2 (0.45) TP53SMN1; SMN2KMT2AMEN1GAA
SCHEMBL9092404 0.63 HRH4 (0.43) HRH4HRH3
SCHEMBL25428682 0.59 TBK1 (0.36) KMT2AMEN1GLAGAA
SCHEMBL9039325 0.59 ALDH1A1 (0.50) MAPTSMN1; SMN2KMT2AGAAHRH4
SCHEMBL21541915 0.57
SCHEMBL30388793 0.56 HRH4 (0.44) MAPTSMN1; SMN2KMT2AMEN1HRH4
SCHEMBL5866936 0.56 KHK (0.46) MAPTSMN1; SMN2KMT2AMEN1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011112731-A2 HETEROCYCLIC INHIBITORS OF HISTAMINE RECEPTORS FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2011-09-15 WO disclosed