SCHEMBL24638845

SCHEMBL24638845

Cc1cncc(C)c1-c1cc(C2CC2)on1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RET P07949 12/20 0.42
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TSHR P16473 1/20 0.39
SMYD3 Q9H7B4 1/20 0.36
CYP1A2 P05177 1/20 0.35
HCK P08631 1/20 0.35
FGR P09769 1/20 0.35
RPS6KB1 P23443 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
MAP2K2 P36507 1/20 0.35
MAP2K1 Q02750 1/20 0.35
RPS6KA1 Q15418 1/20 0.35
S1PR3 Q99500 4/20 0.35
S1PR1 P21453 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24638795 0.83 RET (0.45) RETNPC1RAB9ATSHRCYP1A2
SCHEMBL20952090 0.79 RET (0.41) RETNPC1RAB9ATSHRS1PR3
SCHEMBL17301340 0.73 RAB9A (0.50) RETNPC1RAB9ATSHR
SCHEMBL11836452 0.71 NPC1 (0.45) RETNPC1RAB9ACYP1A2HCK
SCHEMBL28326020 0.71 NPC1 (0.45) RETNPC1RAB9ATSHRSMYD3
SCHEMBL3154169 0.71
SCHEMBL30438396 0.70 RET (0.36) RETNPC1RAB9ATSHRSMYD3
SCHEMBL21530427 0.70 RET (0.43) RETNPC1RAB9ATSHR
SCHEMBL30845491 0.70 RET (0.43) RETNPC1RAB9ATSHR
SCHEMBL11783495 0.69 RAB9A (0.54) RETNPC1RAB9ASMYD3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704114-B1 SPIROCYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2022-11-23 EP disclosed