SCHEMBL24640205

SCHEMBL24640205

CCN1CCN2c3ncc(Cl)c(F)c3OCC2C1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.34
TIPARP Q7Z3E1 1/20 0.34
KRAS P01116 5/20 0.33
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP2D6 P10635 1/20 0.30
LTA4H P09960 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24640610 0.91 TIPARP (0.39) TIPARPKRASHTR2AHTR2CHTR2B
SCHEMBL24639249 0.88 LTA4H (0.33) TIPARPKRASALDH1A1CYP2D6LTA4H
SCHEMBL24639280 0.88 LTA4H (0.33) TIPARPKRASALDH1A1CYP2D6LTA4H
SCHEMBL24640712 0.81 TIPARP (0.34) TIPARPKRAS
SCHEMBL24640214 0.81 TIPARP (0.34) TIPARPKRAS
SCHEMBL24640213 0.81 TIPARP (0.34) TIPARPKRAS
SCHEMBL31244787 0.74 HTR2C (0.49) HTR2AHTR2CHTR2B
SCHEMBL31244708 0.74 HTR2C (0.49) HTR2AHTR2CHTR2B
SCHEMBL24639973 0.72 TIPARP (0.39) TIPARPKRASHTR2AHTR2CHTR2B
SCHEMBL24640609 0.72 TIPARP (0.39) TIPARPKRASHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed