SCHEMBL24639280

SCHEMBL24639280

CCN1CCN2c3ncc(Cl)c(Cl)c3OC[C@H]2C1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.33
KRAS P01116 5/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP2D6 P10635 1/20 0.32
TIPARP Q7Z3E1 1/20 0.32
DRD2 P14416 1/20 0.31
OPRL1 P41146 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639249 1.00 LTA4H (0.33) LTA4HKRASALDH1A1CYP2D6TIPARP
SCHEMBL24640205 0.88 PARP1 (0.34) LTA4HKRASALDH1A1CYP2D6TIPARP
SCHEMBL24640616 0.80 KRAS (0.32) KRASTIPARP
SCHEMBL24640610 0.79 TIPARP (0.39) KRASCYP2D6TIPARPKCNH2
SCHEMBL24639271 0.78 KRAS (0.40) KRASTIPARP
SCHEMBL31245220 0.74 TIPARP (0.48) TIPARP
SCHEMBL24640720 0.72 OPRL1 (0.33) LTA4HOPRL1KCNH2
SCHEMBL24640215 0.71 NLRP3 (0.33) LTA4HOPRL1KCNH2
SCHEMBL24640611 0.70 TIPARP (0.34) KRASTIPARP
SCHEMBL24640207 0.69 TIPARP (0.31) KRASTIPARP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed