SCHEMBL2466067

SCHEMBL2466067

C=CCNCCc1ccc(N(CCC)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 5/20 0.51
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
CNR2 P34972 2/20 0.46
NR3C1 P04150 1/20 0.46
HCRTR2 O43614 1/20 0.46
PTGER1 P34995 1/20 0.41
TRPM8 Q7Z2W7 3/20 0.40
AVPR1B P47901 1/20 0.39
ESR1 P03372 1/20 0.38
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4920488 0.99 SERPINE1 (0.50) SERPINE1LMNAGAAHTTCNR2
SCHEMBL2470902 0.87 HDAC3 (0.49) SERPINE1LMNAGAAHTTCNR2
Hydrochloric Acid SCHEMBL4923250 0.86 HDAC3 (0.48) SERPINE1LMNAGAAHTTCNR2
SCHEMBL2470396 0.82 CNR2 (0.49) CNR2ESR1CNR1
Hydrochloric Acid SCHEMBL4922430 0.81 POLB (0.48) CNR2ESR1CNR1
SCHEMBL2472519 0.77 HDAC1 (0.50) SERPINE1
Hydrochloric Acid SCHEMBL4922816 0.76 HDAC1 (0.49) SERPINE1
SCHEMBL2474733 0.70 HTR6 (0.47) SERPINE1
SCHEMBL7206707 0.68 HDAC1 (0.53)
SCHEMBL5622632 0.68 KEAP1 (0.64) LMNACNR2NR3C1ESR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371814-A1 Aminoethylaromatic compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor Abbott GmbH & Co. KG (DE) 2011-10-05 EP disclosed