SCHEMBL2470396

SCHEMBL2470396

C=CCNCCc1ccc(N(CCC)S(=O)(=O)c2ccc(C(C)C)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.49
CNR1 P21554 7/20 0.49
POLB P06746 1/20 0.49
NPSR1 Q6W5P4 2/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ESR1 P03372 1/20 0.41
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4922430 0.99 POLB (0.48) CNR2CNR1POLBNPSR1TSHR
SCHEMBL2470132 0.86 ALDH1A1 (0.44) CNR2CNR1ALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL4922303 0.85 ALDH1A1 (0.43) CNR2CNR1ALDH1A1MAPTKMT2A
SCHEMBL2466067 0.82 SERPINE1 (0.51) CNR2CNR1ESR1
Hydrochloric Acid SCHEMBL4920488 0.81 SERPINE1 (0.50) CNR2POLBESR1
SCHEMBL1718081 0.78 DRD3 (0.42) POLBALDH1A1MAPTCA12CA1
Hydrochloric Acid SCHEMBL4922945 0.78 DRD3 (0.42) POLBALDH1A1MAPTCA12CA1
SCHEMBL2470496 0.77 ADRB2 (0.57) POLBALDH1A1MAPT
Hydrochloric Acid SCHEMBL4915819 0.76 ADRB2 (0.56) POLBALDH1A1MAPT
SCHEMBL2472844 0.69 CNR2 (0.47) CNR2CNR1POLBNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371814-A1 Aminoethylaromatic compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor Abbott GmbH & Co. KG (DE) 2011-10-05 EP disclosed