SCHEMBL24671531

SCHEMBL24671531

CC(C)(C)OC(=O)N1CC=C(c2ccc(C(=O)Nc3ccc4c(c3)CN(C(=O)OC(C)(C)C)C4)cc2F)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.54
SCN9A Q15858 1/20 0.46
TMPRSS2 O15393 2/20 0.44
PIK3CA P42336 1/20 0.44
MTOR P42345 1/20 0.44
PDK4 Q16654 1/20 0.44
ESR2 Q92731 1/20 0.43
JAK1 P23458 1/20 0.43
NR1H2 P55055 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
GRM5 P41594 3/20 0.42
GRM1 Q13255 3/20 0.42
CDK9 P50750 1/20 0.42
WDR5 P61964 1/20 0.42
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803468 1.00 NAMPT (0.54) NAMPTSCN9ATMPRSS2PIK3CAMTOR
SCHEMBL24670163 0.96 NAMPT (0.51) NAMPTSCN9ATMPRSS2PDK4ESR2
SCHEMBL29803391 0.96 NAMPT (0.51) NAMPTSCN9ATMPRSS2PDK4ESR2
SCHEMBL24669339 0.93 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL29803696 0.93 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670852 0.89 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL29803278 0.89 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24671399 0.89 NAMPT (0.60) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24669383 0.89 NAMPT (0.49) NAMPTSCN9APDK4JAK1NPC1
SCHEMBL24671234 0.89 NAMPT (0.55) NAMPTSCN9ATMPRSS2PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed