SCHEMBL24670320

SCHEMBL24670320

Cc1cc(C2=CCN(/C(=N\C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC2)ccc1C(=O)NC(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.39
SOS1 Q07889 2/20 0.38
CDK7 P50613 1/20 0.36
CDK13 Q14004 1/20 0.36
CDK12 Q9NYV4 1/20 0.36
CCR1 P32246 1/20 0.36
PRMT5 O14744 2/20 0.35
WDR77 Q9BQA1 2/20 0.35
QDPR P09417 2/20 0.35
PDK4 Q16654 1/20 0.34
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
LIPC P11150 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
GRM5 P41594 1/20 0.33
GRM1 Q13255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803536 0.89 NAMPT (0.40) NAMPTSOS1CDK7CDK13CDK12
SCHEMBL24670115 0.88 NAMPT (0.43) NAMPTSOS1CDK7CDK13CDK12
SCHEMBL24891728 0.86 NAMPT (0.46) NAMPT
SCHEMBL29803599 0.86 NAMPT (0.41) NAMPTPRMT5WDR77
SCHEMBL29803471 0.85 NAMPT (0.43) NAMPT
SCHEMBL24669354 0.85 NAMPT (0.42) NAMPTSOS1CDK7CDK13CDK12
SCHEMBL24670906 0.85 NAMPT (0.35) NAMPTSOS1CDK7CDK13CDK12
SCHEMBL24670217 0.85 NAMPT (0.46) NAMPT
SCHEMBL24671366 0.85 NAMPT (0.39) NAMPTSOS1CDK7CDK13CDK12
SCHEMBL24670218 0.85 NAMPT (0.46) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed