SCHEMBL24670475

SCHEMBL24670475

N=C(N)N1CC=C(c2ccc(NC(=O)c3cnc(C4=CCN(C(=N)N)CC4)s3)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.46
PTPN1 P18031 1/20 0.45
NAMPT P43490 16/20 0.43
NPC1 O15118 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ALOX15 P16050 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 1/20 0.42
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29803352 0.93 PTPN11 (0.43) PTPN11PTPN1NAMPTNPC1ALDH1A1
SCHEMBL29802997 0.88 PTPN11 (0.39) PTPN11PTPN1NAMPTMAPT
SCHEMBL29803304 0.86 HDAC2 (0.45) NAMPTNPC1ALDH1A1ALOX15RAB9A
SCHEMBL24671076 0.86 PTPN11 (0.38) PTPN11PTPN1NAMPT
Hydrochloric Acid SCHEMBL29803300 0.85 HDAC2 (0.44) NAMPTNPC1ALDH1A1ALOX15RAB9A
SCHEMBL29803084 0.83 ESRRG (0.46) PTPN11PTPN1NAMPTNPC1ALDH1A1
SCHEMBL24669181 0.82 NAMPT (0.61) PTPN1NAMPTSMN1; SMN2TSHRMAPT
Trifluoroacetic Acid SCHEMBL29803396 0.81 TRPV1 (0.38) PTPN11PTPN1
SCHEMBL24667821 0.81 TMPRSS2 (0.54) NAMPTNPC1ALDH1A1ALOX15RAB9A
SCHEMBL24669917 0.81 ALDH1A1 (0.44) NAMPTNPC1ALDH1A1ALOX15RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO claimed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed