SCHEMBL24671076

SCHEMBL24671076

N=C(N)NCCc1ccc(NC(=O)c2cnc(C3=CCN(C(=N)N)CC3)s2)cc1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.38
PTPN1 P18031 1/20 0.37
TRPV1 Q8NER1 7/20 0.36
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
JAK1 P23458 2/20 0.35
TMPRSS2 O15393 2/20 0.35
JAK2 O60674 1/20 0.35
NAMPT P43490 4/20 0.34
EGLN1 Q9GZT9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29803396 0.94 TRPV1 (0.38) PTPN11PTPN1TRPV1EGLN1
SCHEMBL29802997 0.91 PTPN11 (0.39) PTPN11PTPN1TRPV1SLC6A3KCNH2
SCHEMBL24670475 0.86 PTPN11 (0.46) PTPN11PTPN1NAMPT
SCHEMBL24670463 0.84 PTPN11 (0.40) PTPN11PTPN1TRPV1SLC6A3KCNH2
SCHEMBL24671165 0.82 ALDH1A1 (0.36) TMPRSS2NAMPTEGLN1
SCHEMBL24670895 0.82 TMPRSS2 (0.44) JAK1TMPRSS2JAK2NAMPT
Trifluoroacetic Acid SCHEMBL29803352 0.80 PTPN11 (0.43) PTPN11PTPN1TRPV1NAMPTEGLN1
SCHEMBL24671416 0.80 TP53 (0.37) TMPRSS2NAMPT
SCHEMBL24669205 0.80 MAPT (0.36) TMPRSS2NAMPT
SCHEMBL24670472 0.79 NAMPT (0.49) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO claimed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed