SCHEMBL24670643

SCHEMBL24670643

N=C(N)N1CC=C(c2ccc(C(=O)Nc3ccc(C4=CCN(C(=N)N)CC4)c(Cl)c3)cc2F)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 6/20 0.52
MAPT P10636 5/20 0.45
LMNA P02545 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HTT P42858 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CHRM1 P11229 1/20 0.42
TRPV1 Q8NER1 5/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29802861 1.00 TMPRSS2 (0.52) TMPRSS2MAPTLMNAMEN1KMT2A
SCHEMBL29803214 0.93 TMPRSS2 (0.52) TMPRSS2MAPTLMNATRPV1NPC1
SCHEMBL29802931 0.93 TMPRSS2 (0.59) TMPRSS2MAPTLMNAMEN1KMT2A
SCHEMBL24670920 0.91 CHRM1 (0.53) TMPRSS2MAPTLMNAMEN1KMT2A
SCHEMBL24669447 0.89 TMPRSS2 (0.48) TMPRSS2MAPTLMNAHTTALDH1A1
SCHEMBL24671270 0.89 TMPRSS2 (0.52) TMPRSS2MAPTLMNAMEN1KMT2A
SCHEMBL29803204 0.89 TMPRSS2 (0.52) TMPRSS2MAPTLMNAMEN1KMT2A
SCHEMBL29802975 0.88 TMPRSS2 (0.59) TMPRSS2NPC1
SCHEMBL24670135 0.88 TMPRSS2 (0.59) TMPRSS2NPC1
SCHEMBL24671177 0.87 TMPRSS2 (0.51) TMPRSS2MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed