SCHEMBL24670832

SCHEMBL24670832

COc1cc(NC(=O)c2ccc(C3=CCN(C=NC(=O)OC(C)(C)C)CC3)c(Cl)c2)ccc1C1=CCN(C(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
NAMPT P43490 5/20 0.35
MAOB P27338 1/20 0.34
ROCK2 O75116 1/20 0.34
ABCB1 P08183 2/20 0.33
NPC1 O15118 1/20 0.33
MCHR1 Q99705 1/20 0.33
ATM Q13315 1/20 0.33
APOBEC3G Q9HC16 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670867 0.94 MAPT (0.39) MAPTTP53THRBSMN1; SMN2TRPV1
SCHEMBL24670860 0.94 MAPT (0.39) MAPTTP53THRBSMN1; SMN2TRPV1
SCHEMBL24671510 0.93 NAMPT (0.41) NAMPTABCB1MCHR1
SCHEMBL24670242 0.90 NPC1 (0.35) TRPV1NAMPTABCB1NPC1MCHR1
SCHEMBL29803748 0.89 NAMPT (0.40) MAPTTP53THRBSMN1; SMN2TRPV1
SCHEMBL24670803 0.88 NAMPT (0.38) MAPTTP53SMN1; SMN2NAMPTABCB1
SCHEMBL24670937 0.88 NAMPT (0.34) MAPTTRPV1NAMPTABCB1NPC1
SCHEMBL24671554 0.88 NAMPT (0.34) MAPTSMN1; SMN2TRPV1NAMPTABCB1
SCHEMBL24670776 0.86 HTR1D (0.38) MAPTSMN1; SMN2NAMPTROCK2ABCB1
SCHEMBL24670811 0.86 TRPV1 (0.39) MAPTTP53SMN1; SMN2TRPV1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed