SCHEMBL24670937

SCHEMBL24670937

COc1cc(NC(=O)c2ccc(C3=CCN(C=NC(=O)OC(C)(C)C)CC3)c(F)c2F)ccc1C1=CCN(C(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.34
TRPV1 Q8NER1 2/20 0.34
CCNT1 O60563 2/20 0.32
CDK9 P50750 2/20 0.32
ABCB1 P08183 2/20 0.32
GRM5 P41594 1/20 0.32
GRM1 Q13255 1/20 0.32
MTTP P55157 3/20 0.31
NPC1 O15118 1/20 0.31
AVPR2 P30518 1/20 0.31
AVPR1A P37288 1/20 0.31
AVPR1B P47901 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
RECQL P46063 1/20 0.31
CHRNA1 P02708 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CHRNB2 P17787 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670707 0.93 TRPV1 (0.36) NAMPTTRPV1CCNT1CDK9GRM5
SCHEMBL24670703 0.93 TRPV1 (0.36) NAMPTTRPV1CCNT1CDK9GRM5
SCHEMBL24671259 0.92 NAMPT (0.38) NAMPTTRPV1ABCB1MTTPNPC1
SCHEMBL24671554 0.92 NAMPT (0.34) NAMPTTRPV1CCNT1CDK9ABCB1
SCHEMBL24670803 0.90 NAMPT (0.38) NAMPTABCB1KDM4EMAPTCYP3A4
SCHEMBL24670242 0.90 NPC1 (0.35) NAMPTTRPV1CCNT1CDK9ABCB1
SCHEMBL24671510 0.89 NAMPT (0.41) NAMPTABCB1
SCHEMBL24670832 0.88 MAPT (0.37) NAMPTTRPV1ABCB1NPC1MAPT
SCHEMBL24670926 0.84 WDR5 (0.36) NAMPTTRPV1CCNT1CDK9NPC1
SCHEMBL24671551 0.84 WDR5 (0.36) NAMPTTRPV1CCNT1CDK9NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed