SCHEMBL24671042

SCHEMBL24671042

CCc1ccc(C(=N)c2c(N)ncnc2NC(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.36
SRC P12931 2/20 0.35
EGFR P00533 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PIK3CD O00329 2/20 0.32
F7 P08709 1/20 0.32
BTK Q06187 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
SYK P43405 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPT P10636 1/20 0.32
DGAT1 O75907 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
PKM P14618 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PRMT1 Q99873 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671954 0.80 SRC (0.40) SRCSMN1; SMN2PIK3CDBTKLMNA
SCHEMBL13430257 0.77 SRC (0.54) SRCEGFRSMN1; SMN2SYKMAPT
SCHEMBL24862167 0.75 EGFR (0.53) EGFRBTKHPGD
SCHEMBL21082555 0.75 SRC (0.35) SRCSMN1; SMN2PIK3CDLMNAHTT
SCHEMBL23287652 0.75 PIK3CD (0.47) SRCSMN1; SMN2PIK3CDALDH1A1HPGD
SCHEMBL18518847 0.75 RET (0.39) SRCSMN1; SMN2PIK3CDALDH1A1HPGD
SCHEMBL21501448 0.75 PIK3CA (0.45) SRCPIK3CDCYP1A2MAPTLMNA
SCHEMBL18518829 0.74 SMN1; SMN2 (0.39) SRCSMN1; SMN2PIK3CDALDH1A1HPGD
SCHEMBL22539865 0.74 PIK3CA (0.42) SRCSMN1; SMN2PIK3CDCYP3A4LMNA
SCHEMBL8008751 0.74 ALDH1A1 (0.42) CYP2C19SMN1; SMN2PIK3CDALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4043465-A1 SUBSTITUTED AROMATIC FUSED RING DERIVATIVE AND COMPOSITION COMPRISING SAME, AND USE THEREOF Shenzhen TargetRx, Inc. (CN) 2022-08-17 EP disclosed