SCHEMBL24671051

SCHEMBL24671051

CC(C)(C)OC(=O)NCCc1ccc(NC(=O)c2cc(Br)cs2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.52
HRH3 Q9Y5N1 6/20 0.46
FPR2 P25090 6/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
PTGER4 P35408 1/20 0.42
FPR3 P25089 5/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LEF1 Q9UJU2 1/20 0.41
CNR1 P21554 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669864 0.89 NAMPT (0.50) NAMPTFPR2FPR3HDAC1HDAC6
SCHEMBL24669430 0.82 NAMPT (0.55) NAMPTFPR2CA1CA2FPR3
SCHEMBL24669866 0.82 NAMPT (0.51) NAMPTFPR2CA1CA2PTGER4
SCHEMBL24670295 0.79 RAB9A (0.53) NAMPTFPR2CA1CA2FPR3
SCHEMBL24671047 0.79 RAB9A (0.56) NAMPTLMNAALDH1A1
SCHEMBL1065312 0.78 CA2 (0.55) NAMPTFPR2CA1CA2FPR3
SCHEMBL2873843 0.77 NAMPT (0.64) NAMPTHDAC1
SCHEMBL24669863 0.77 NAMPT (0.53) NAMPTCA1CA2LMNAALDH1A1
SCHEMBL29803548 0.77 NAMPT (0.53) NAMPTCA1CA2LMNAALDH1A1
SCHEMBL19889037 0.77 NAMPT (0.60) NAMPTFPR2CA1CA2FPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed