SCHEMBL24671182

SCHEMBL24671182

COc1cc(NC(=O)c2ccc(C3=CCN(C(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC3)c(F)c2)ccc1C1=CCN(C(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.38
NPC1 O15118 3/20 0.38
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
SCN9A Q15858 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ABCB1 P08183 2/20 0.35
TRPV1 Q8NER1 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
KMT2A Q03164 1/20 0.35
TMPRSS2 O15393 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803596 1.00 NAMPT (0.38) NAMPTNPC1KCNQ3KCNQ2CCNT1
SCHEMBL29803193 0.95 NAMPT (0.40) NAMPTNPC1CDK9SCN9ATP53
SCHEMBL29803771 0.93 TRPV1 (0.39) NAMPTSCN9ATRPV1
SCHEMBL24670267 0.93 TRPV1 (0.39) NAMPTSCN9ATRPV1
SCHEMBL24671542 0.93 CDK9 (0.36) NAMPTNPC1CCNT1CDK9MAPT
SCHEMBL24670237 0.93 CDK9 (0.36) NAMPTNPC1CCNT1CDK9MAPT
SCHEMBL24671294 0.93 MAPT (0.37) NAMPTNPC1TP53MAPTTHRB
SCHEMBL24671296 0.93 MAPT (0.37) NAMPTNPC1TP53MAPTTHRB
SCHEMBL24669443 0.93 KCNQ3 (0.38) NAMPTNPC1KCNQ3KCNQ2CCNT1
SCHEMBL24669449 0.93 KCNQ3 (0.38) NAMPTNPC1KCNQ3KCNQ2CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed