SCHEMBL24671229

SCHEMBL24671229

CCc1ccc(NC(=O)c2cnc(C3=CCN(C(=O)OC(C)(C)C)CC3)s2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.51
WNT3A P56704 1/20 0.48
GPR119 Q8TDV5 2/20 0.45
GRM1 Q13255 4/20 0.43
GRM5 P41594 3/20 0.43
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KIT P10721 1/20 0.41
PDK4 Q16654 1/20 0.41
TP53 P04637 1/20 0.41
EED O75530 2/20 0.41
RBBP4 Q09028 2/20 0.41
SUZ12 Q15022 2/20 0.41
EZH2 Q15910 2/20 0.41
SCN9A Q15858 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669181 0.91 NAMPT (0.61) NAMPTWNT3AGPR119GRM1GRM5
SCHEMBL29803758 0.90 NAMPT (0.48) NAMPTWNT3AGPR119GRM1GRM5
SCHEMBL24670472 0.88 NAMPT (0.49) NAMPTWNT3AGPR119GRM1GRM5
SCHEMBL31705574 0.82 GPR119 (0.48) NAMPTGPR119GRM1GRM5PDK4
SCHEMBL31705452 0.82 GPR119 (0.48) NAMPTGPR119GRM1GRM5PDK4
SCHEMBL24669894 0.78 HDAC3 (0.40) NAMPTWNT3AMAPTKITHDAC3
SCHEMBL29803417 0.78 HDAC3 (0.40) NAMPTWNT3AMAPTKITHDAC3
SCHEMBL24670464 0.78 HDAC3 (0.40) NAMPTWNT3AMAPTKITHDAC3
SCHEMBL29803354 0.77 HDAC3 (0.41) NAMPTWNT3AHDAC3HDAC4HDAC1
SCHEMBL23164675 0.77 NAMPT (0.49) NAMPTWNT3AGPR119GRM1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed