SCHEMBL24671309

SCHEMBL24671309

COCNc1cc(F)c(C2=CCN(C(=O)OC(C)(C)C)CC2)cc1C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.46
GRM5 P41594 7/20 0.45
GRM1 Q13255 7/20 0.45
WDR5 P61964 2/20 0.44
JAK1 P23458 1/20 0.44
CDK9 P50750 3/20 0.42
CCNT1 O60563 1/20 0.42
NAMPT P43490 1/20 0.41
HTR6 P50406 1/20 0.41
EED O75530 2/20 0.40
RBBP4 Q09028 2/20 0.40
SUZ12 Q15022 2/20 0.40
EZH2 Q15910 2/20 0.40
TNF P01375 1/20 0.40
SCN9A Q15858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670885 0.87 CDK9 (0.51) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24670170 0.83 WDR5 (0.53) PDK4GRM5GRM1WDR5JAK1
SCHEMBL29803388 0.83 WDR5 (0.53) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24718042 0.82 PDK4 (0.48) PDK4GRM5GRM1WDR5JAK1
SCHEMBL30798488 0.82 PDK4 (0.48) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24670953 0.81 PDK4 (0.51) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24669316 0.80 WDR5 (0.48) PDK4GRM5GRM1WDR5JAK1
SCHEMBL29803452 0.80 WDR5 (0.48) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24670313 0.80 NAMPT (0.49) PDK4GRM5GRM1WDR5JAK1
SCHEMBL24671112 0.78 WDR5 (0.49) PDK4GRM5GRM1WDR5JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed