SCHEMBL24671357

SCHEMBL24671357

CCc1cc(C2=CCN(C(N)N)CC2)ccc1C(=O)Nc1ccc(C2=CCN(C(=N)N)CC2)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.36
MMP3 P08254 2/20 0.36
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PLG P00747 1/20 0.35
PLAU P00749 1/20 0.35
PLAT P00750 1/20 0.35
NAMPT P43490 6/20 0.35
TMPRSS2 O15393 2/20 0.35
HTR1D P28221 3/20 0.35
HTR1B P28222 3/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671362 0.94 MMP2 (0.40) MMP2MMP3F2F10PLG
SCHEMBL24671333 0.84 MAPT (0.41) MMP2MMP3F2F10PLG
SCHEMBL24671353 0.84 TMPRSS2 (0.43) MMP2MMP3F2F10PLG
SCHEMBL24670308 0.81 TRPV1 (0.45) MMP2MMP3NAMPTMAPTLMNA
SCHEMBL29803440 0.80 NAMPT (0.50) NAMPT
SCHEMBL24669458 0.78 TMPRSS2 (0.48) F2PLGPLAUPLATNAMPT
SCHEMBL24670299 0.77 MAPT (0.46) MMP2MMP3NAMPTTMPRSS2MAPT
SCHEMBL24671261 0.77 QDPR (0.43) PLAUPLATNAMPTTMPRSS2HTR1D
SCHEMBL24669447 0.76 TMPRSS2 (0.48) NAMPTTMPRSS2MAPTLMNAHTT
SCHEMBL29803214 0.76 TMPRSS2 (0.52) PLAUNAMPTTMPRSS2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed