SCHEMBL24672721

SCHEMBL24672721

N=Cc1c(NC[C@H]2OC(O)[C@@H](O)C2=O)nc(Cl)nc1NC1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.36
ADORA1 P30542 7/20 0.36
ADORA2A P29274 6/20 0.36
ADORA2B P29275 4/20 0.36
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
NT5E P21589 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19822682 0.64 KMT2A (0.36) ADORA3ADORA1ADORA2AKMT2A
SCHEMBL23599060 0.61 CA1 (0.54)
SCHEMBL19659465 0.57 KMT2A (0.64) ADORA3ADORA1ADORA2AADORA2BMEN1
SCHEMBL8334814 0.56 PDE9A (0.43) ADORA1ADORA2AADORA2BMEN1CYP1A2
SCHEMBL20776751 0.56 YTHDC1 (0.34) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL30956669 0.56 KMT2A (0.38) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL22412912 0.56 KMT2A (0.38) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL22411428 0.55 KMT2A (0.40) ADORA3ADORA1ADORA2AADORA2BMEN1
SCHEMBL30873856 0.55 KMT2A (0.40) ADORA3ADORA1ADORA2AADORA2BMEN1
SCHEMBL14196007 0.54 IRAK4 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237747-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF 四川海思科制药有限公司 2022-11-17 WO disclosed