SCHEMBL24674717

SCHEMBL24674717

CC(C)(C)OC(=O)N1CCN(c2ncc(C(F)(F)F)cc2Br)[C@H](CO)C1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CXCR3 P49682 1/20 0.41
HDAC6 Q9UBN7 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
GPR119 Q8TDV5 8/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.37
MDM2 Q00987 1/20 0.37
TACR1 P25103 1/20 0.37
STS P08842 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24763856 1.00 MEN1 (0.42) MEN1KMT2ACXCR3HDAC6HDAC8
SCHEMBL24675006 0.91 MEN1 (0.41) MEN1KMT2AHDAC6HDAC8GPR119
SCHEMBL30658110 0.91 MEN1 (0.41) MEN1KMT2AHDAC6HDAC8GPR119
SCHEMBL30729623 0.90 CXCR3 (0.50) MEN1KMT2ACXCR3HDAC6GPR119
SCHEMBL31491286 0.90 CXCR3 (0.50) MEN1KMT2ACXCR3HDAC6GPR119
SCHEMBL26958997 0.90 CXCR3 (0.50) MEN1KMT2ACXCR3HDAC6GPR119
SCHEMBL14465886 0.90 CXCR3 (0.50) MEN1KMT2ACXCR3HDAC6GPR119
SCHEMBL24764604 0.88 GPR119 (0.42) HDAC6HDAC8GPR119
SCHEMBL24675003 0.88 HDAC6 (0.40) MEN1KMT2AHDAC6HDAC8GPR119
SCHEMBL29274215 0.88 HDAC6 (0.40) MEN1KMT2AHDAC6HDAC8GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117083274-A Fused ring heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2023-11-17 CN disclosed
WO-2022223022-A1 FUSED-RING HETEROCYCLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 四川海思科制药有限公司 2022-10-27 WO disclosed