SCHEMBL24675993

SCHEMBL24675993

Cc1nc(N(CCN(C)C)C(=O)OC(C)(C)C)sc1-c1cc(Cl)ncc1C#N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RAB9A P51151 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
POLB P06746 1/20 0.32
GLA P06280 1/20 0.32
USP7 Q93009 1/20 0.32
USP47 Q96K76 1/20 0.32
AAK1 Q2M2I8 2/20 0.31
RET P07949 2/20 0.31
HTR2C P28335 1/20 0.31
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30
RAD52 P43351 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676006 0.76 GPBAR1 (0.34) NR1H2NR1H3
SCHEMBL29755073 0.76 GPBAR1 (0.34) NR1H2NR1H3
SCHEMBL28511505 0.70 ADORA2A (0.37) ALDH1A1GLA
SCHEMBL24675926 0.70 CA12 (0.35) ALDH1A1SMN1; SMN2LMNAMAPK1MAPT
SCHEMBL30756386 0.67 AAK1 (0.36) ALDH1A1LMNAKMT2AGLAAAK1
SCHEMBL24676814 0.66 AAK1 (0.39) AAK1HTR2C
SCHEMBL30907180 0.61 SYK (0.34) AAK1
SCHEMBL30926187 0.61 STK17B (0.36) ALDH1A1
SCHEMBL19675997 0.61 CA12 (0.35) AAK1
SCHEMBL19020601 0.61 RET (0.37) RETNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed