SCHEMBL24676771

SCHEMBL24676771

CCc1nc(O)ccc1C(=O)c1c(CC)oc2cc(C#N)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 11/20 0.46
TTR P02766 4/20 0.43
EYA3 Q99504 6/20 0.43
CYP2C19 P33261 6/20 0.41
CYP2C9 P11712 2/20 0.39
MEN1 O00255 2/20 0.39
ABCB11 O95342 2/20 0.39
LMNA P02545 2/20 0.39
PGR P06401 2/20 0.39
ADRA2A P08913 2/20 0.39
TBXA2R P21731 2/20 0.39
OPRM1 P35372 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KMT2A Q03164 2/20 0.39
BIRC5 O15392 1/20 0.39
HTR1A P08908 1/20 0.39
DRD1 P21728 1/20 0.39
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
PDE4A P27815 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20366740 0.71 ALK (0.41) SLC22A12TTREYA3CYP3A4MAPT
SCHEMBL1287582 0.68 EYA3 (0.71) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL20004875 0.65 GSK3B (0.35) MEN1KMT2A
SCHEMBL1287413 0.64 SLC22A12 (1.00) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL28104862 0.64 EYA3 (0.57) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL29286599 0.63 EYA3 (0.70) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL6338104 0.62 EYA3 (0.70) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL28104498 0.62 EYA3 (0.64) SLC22A12TTREYA3CYP2C19CYP2C9
SCHEMBL7449274 0.61 HSD17B3 (0.44) ALDH1A1
SCHEMBL9444753 0.61 EYA3 (0.68) SLC22A12TTREYA3CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230142119-A1 TETRACYCLIC COMPOUND CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-05-11 US disclosed
US-20220306578-A1 TETRACYCLIC COMPOUND CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2022-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230142119-A1 TETRACYCLIC COMPOUND ALK, TTR, ACVR1 SLC22A12 1472/4885TTR 2/4885EYA3 1232/4885
US-20220306578-A1 TETRACYCLIC COMPOUND ALK, TTR, ACVR1 SLC22A12 1472/4885TTR 2/4885EYA3 1232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.