Tecadenoson

Tecadenoson

SCHEMBL246787

OC[C@H]1O[C@@H](n2cnc3c(N[C@@H]4CCOC4)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1

The experimentally established mechanism targets of Tecadenoson. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 known ✓ P30542 9/20 1.00
ADORA2A P29274 7/20 1.00
ADORA3 P0DMS8 7/20 1.00
ADORA2B P29275 4/20 1.00
SLC29A1 Q99808 2/20 1.00
SLC28A1 O00337 1/20 1.00
TSHR P16473 3/20 0.78
PMP22 Q01453 2/20 0.78
GAA P10253 1/20 0.78
HTT P42858 1/20 0.78
SIGMAR1 Q99720 1/20 0.78
RXFP1 Q9HBX9 1/20 0.78
MEN1 O00255 1/20 0.78
KMT2A Q03164 1/20 0.78
TP53 P04637 1/20 0.78
NFKB1 P19838 1/20 0.78
HIF1A Q16665 1/20 0.78
SMN1; SMN2 Q16637 1/20 0.77
TDP1 Q9NUW8 1/20 0.77
CYP2C19 P33261 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tecadenoson SCHEMBL15106888 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL472425 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL1095647 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL472549 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL15106884 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL12265126 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL24838611 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL6226634 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL22349437 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1
Tecadenoson SCHEMBL7034923 1.00 ADORA1 (1.00) ADORA1ADORA2AADORA3ADORA2BSLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 418 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2026-05-28 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20240139325-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2024-05-02 US claimed
EP-4178948-A2 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF Universidade de Santiago de Compostela (ES) 2023-05-17 EP claimed
EP-4045504-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS Ai-biopharma (FR) 2022-08-24 EP claimed
CN-114376962-A Drug-loaded nanofiber for acupuncture point thread embedding material and preparation method and application thereof 上海市第四人民医院 2022-04-22 CN claimed
WO-2022023496-A2 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2022-02-03 WO claimed
WO-2021074443-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2021-04-22 WO claimed
US-20200276312-A1 Elimination of chronic pain by chronic activation of adenosine receptor type A1 in peripheral sensory neurons UNIV ROCHESTER (US) 2020-09-03 US claimed
WO-2019178267-A2 INDUCTIVE REGENERATION OF THE AIRWAY BY TRANSCRIPTIONAL FACTOR MODULATION OF GLANDULAR MYOEPITHELIAL STEM CELLS UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2019-09-19 WO claimed
WO-2008063323-A2 TREATMENT WITH ANTIARRHYTHMICS AND OMEGA-3 FATTY ACIDS AND A COMBINATION PRODUCT THEREOF RELIANT PHARMACEUTICALS, INC. (US) 2008-05-29 WO claimed
WO-2007073855-A1 USE OF ADENOSINE A1 RECEPTOR AGONISTS FOR THE PROTECTION OF RENAL CELLS AGAINST TOXIC EFFECTS CAUSED BY AMINOGLYCOSIDES DURING TREATMENT OF INFECTIOUS DISEASES BAYER HEALTHCARE AG (DE) 2007-07-05 WO claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20050074425-A1 Method for delivering polymerized therapeutic agent compositions and compositions thereof POLYCORD, INC. (US) 2005-04-07 US claimed
WO-2005002597-A1 METHOD FOR DELIVERING POLYMERIZED THERAPEUTIC AGENT COMPOSITIONS AND COMPOSITIONS THEREOF POLYCORD, INC. (US) 2005-01-13 WO claimed
WO-2004056181-A1 ORGAN PRECONDITIONING, ARREST, PROTECTION, PRESERVATION AND RECOVERY (2) GLOBAL CARDIAC SOLUTIONS PTY LTD (AU) 2004-07-08 WO claimed
WO-2004056180-A1 ORGAN PRECONDITIONING, ARREST, PROTECTION, PRESERVATION AND RECOVERY (1) GLOBAL CARDIAC SOLUTIONS PTY LTD (AU) 2004-07-08 WO claimed
EP-0992510-B1 N6 heterocyclic substituted adenosine derivatives CV THERAPEUTICS INC (US) 2003-03-12 EP claimed
US-20020037871-A1 Pharmaceutical use of adenosine agonists CAN-FITE BIOPHARMA LTD. (IL) 2002-03-28 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS HAVCR2, NR1H4, NR1H3 ADORA1 515/4885ADORA2A 1902/4885ADORA3 558/4885
US-20020037871-A1 Pharmaceutical use of adenosine agonists ADORA1, ADORA2A, ADORA3 ADORA1 1/4885ADORA2A 2/4885ADORA3 3/4885
US-20240139325-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS SLC10A1, HAVCR2, HDGF ADORA1 4210/4885ADORA2A 4586/4885ADORA3 3777/4885
US-20200276312-A1 Elimination of chronic pain by chronic activation of adenosine receptor type A1 in peripheral sensory neurons P2RX3, P2RX1, P2RX2 ADORA1 4/4885ADORA2A 8/4885ADORA3 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.