SCHEMBL2468153

SCHEMBL2468153

COc1cc(OC)cc(C(O)C#Cc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.51
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
NLRP3 Q96P20 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
IDO1 P14902 1/20 0.38
HSD17B2 P37059 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2E1 P05181 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2802710 0.88 AOC3 (0.46) DHFRHSD17B2
SCHEMBL13859211 0.87 DHFR (0.45) DHFRMEN1KMT2APDE4APDE4B
SCHEMBL22122696 0.85 KMT2A (0.47) DHFRMEN1KMT2ANPC1POLB
SCHEMBL2683955 0.85 KMT2A (0.47) DHFRMEN1KMT2ANPC1POLB
SCHEMBL2466860 0.84 DHFR (0.39) DHFRIDO1
SCHEMBL23572596 0.82 APP (0.49) DHFRMEN1KMT2ANPC1POLB
SCHEMBL2685285 0.82 APP (0.49) DHFRMEN1KMT2ANPC1POLB
SCHEMBL2519799 0.77 TSHR (0.52) KMT2APOLBIDO1CYP1A2CYP3A4
SCHEMBL2801832 0.77 TSHR (0.52) KMT2APOLBIDO1CYP1A2CYP3A4
SCHEMBL17845069 0.77 APP (0.48) KMT2APOLBIDO1HSD17B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119778-A2 METHOD FOR IN-SITU FORMATION OF METATHESIS CATALYSTS SCHRODI YANN (US) 2011-09-29 WO disclosed