SCHEMBL24684142

SCHEMBL24684142

NC(=O)c1ccc(NC(=O)c2cc(C(F)(F)F)cnc2Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 4/20 0.51
ATF1 P18846 2/20 0.51
KCNQ3 O43525 2/20 0.50
KCNQ2 O43526 2/20 0.50
KCNE1 P15382 2/20 0.50
KCNQ1 P51787 2/20 0.50
SCN10A Q9Y5Y9 2/20 0.49
P2RY14 Q15391 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
TYK2 P29597 1/20 0.48
BCAT2 O15382 1/20 0.48
KIT P10721 1/20 0.47
MAPT P10636 2/20 0.47
JUN P05412 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
SORT1 Q99523 1/20 0.46
P2RX1 P51575 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29804497 0.87 PTGES (0.52) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL24682601 0.87 PTGES (0.52) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL1585024 0.86 NFKB1 (0.52) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL28049181 0.83 KCNQ3 (0.50) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL21906016 0.82 SCN10A (0.68) SCN10AJAK2JAK1TYK2SORT1
SCHEMBL28049179 0.81 KCNQ3 (0.48) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL29732883 0.80 P2RX1 (0.60) KCNQ3KCNQ2KCNE1KCNQ1SMN1; SMN2
SCHEMBL28789750 0.80 P2RX1 (0.60) KCNQ3KCNQ2KCNE1KCNQ1SMN1; SMN2
SCHEMBL5414532 0.80 P2RX1 (0.64) NFKB1ATF1KCNQ3KCNQ2KCNE1
SCHEMBL22435417 0.79 CYP1A2 (0.50) NFKB1ATF1KITJUNNFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240336574-A1 METHYL-SUBSTITUTED PYRIDINE AND PYRIDAZINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. 2024-10-10 US disclosed
EP-4304585-A2 METHYL-SUBSTITUTED PYRIDINE AND PYRIDAZINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE Latigo Biotherapeutics, Inc. (US) 2024-01-17 EP disclosed
CN-117062607-A Methyl substituted pyridine and pyridazine compounds, derivatives thereof and methods of use thereof 拉堤果生物医疗股份有限公司 2023-11-14 CN disclosed
WO-2022192487-A2 METHYL-SUBSTITUTED PYRIDINE AND PYRIDAZINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. (US) 2022-09-15 WO disclosed
WO-2022192487-A2 METHYL-SUBSTITUTED PYRIDINE AND PYRIDAZINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. (US) 2022-09-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240336574-A1 METHYL-SUBSTITUTED PYRIDINE AND PYRIDAZINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE P2RX5, HRH4, TRPV1 NFKB1 1918/4885ATF1 1889/4885KCNQ3 939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.