SCHEMBL2469685

SCHEMBL2469685

C#Cc1ccc(NC(=O)O)c(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.40
GAA P10253 7/20 0.38
KDM4E B2RXH2 6/20 0.38
ALDH1A1 P00352 4/20 0.38
MAP2K2 P36507 1/20 0.38
MAP2K1 Q02750 1/20 0.38
MAPT P10636 5/20 0.36
THRB P10828 3/20 0.36
HPGD P15428 3/20 0.36
GFER P55789 3/20 0.36
HSD17B10 Q99714 3/20 0.36
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GLA P06280 1/20 0.36
RCE1 Q9Y256 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18493542 0.84 HPGD (0.39) MAP2K2MAP2K1HPGDNPC1CYP2C9
SCHEMBL2134811 0.77 AAK1 (0.44)
SCHEMBL2465151 0.76 GABRA1 (0.36) HDAC1GAAKDM4EALDH1A1MAPT
SCHEMBL6609844 0.74 ALDH1A1 (0.47) ALDH1A1MAPTNPC1SMN1; SMN2GLA
SCHEMBL15009906 0.74 SMN1; SMN2 (0.50) HDAC1GAAKDM4EALDH1A1MAPT
SCHEMBL1266865 0.73 HDAC1 (0.68) HDAC1ALDH1A1NPC1SMN1; SMN2HDAC3
SCHEMBL15559293 0.73 AAK1 (0.55) HDAC1KDM4EALDH1A1MAPTNPC1
SCHEMBL21857320 0.73 ALDH1A1 (0.49) GAAKDM4EALDH1A1MAPTTHRB
SCHEMBL3953891 0.73 HDAC1 (0.55) HDAC1GAAKDM4EALDH1A1HPGD
SCHEMBL978331 0.72 GAA (0.49) HDAC1GAAKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367599-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY Massachusetts Institute of Technology (US) 2011-09-28 EP disclosed
WO-2010065117-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-06-10 WO disclosed