SCHEMBL24697142

SCHEMBL24697142

c1ccc(CN2CC[C@@H]2c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.49
TP53 P04637 1/20 0.49
MDM2 Q00987 1/20 0.49
SIGMAR1 Q99720 6/20 0.47
ACHE P22303 1/20 0.46
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
CCR3 P51677 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2172790 0.89 CHRNB2 (0.53) TP53MDM2
SCHEMBL22201130 0.89 CHRNB2 (0.53) TP53MDM2
SCHEMBL11488897 0.87 KDM4E (0.56)
SCHEMBL24365232 0.87 KDM4E (0.56)
SCHEMBL537320 0.83 SIGMAR1 (0.49) GBA1TP53MDM2SIGMAR1ACHE
SCHEMBL6269988 0.83 SIGMAR1 (0.53) GBA1TP53MDM2SIGMAR1NR1H2
SCHEMBL23064631 0.80 MEN1 (0.55) SIGMAR1
SCHEMBL23064641 0.80 DRD2 (0.54) SIGMAR1
SCHEMBL16226782 0.79 SIGMAR1 (0.55) TP53MDM2SIGMAR1NR1H2NR1H3
SCHEMBL9070276 0.79 DRD2 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3412663-B1 NITROGEN-CONTAINING HETEROCYCLE AND CARBOCYCLE DERIVATIVES HAVING TRKA INHIBITORY ACTIVITY SHIONOGI & CO (JP) 2022-09-07 EP disclosed