SCHEMBL24697343

SCHEMBL24697343

CCc1cccc2cc(O)cc(N)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.44
GABRB2 P47870 2/20 0.44
DAO P14920 2/20 0.41
ELANE P08246 2/20 0.40
FLT3 P36888 1/20 0.39
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ANPEP P15144 1/20 0.36
DPP4 P27487 1/20 0.36
KRAS P01116 1/20 0.34
PARP1 P09874 1/20 0.34
DDO Q99489 1/20 0.34
TLR8 Q9NR97 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MTNR1A P48039 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24630603 0.84 GABRA1 (0.48) GABRA1GABRB2DAOELANEFLT3
SCHEMBL25811575 0.83 ALDH1A1 (0.33) ALDH1A1
SCHEMBL24175936 0.81 GABRA1 (0.45) GABRA1GABRB2DAOELANEFLT3
SCHEMBL25811635 0.80 HTR2A (0.34) ALDH1A1HTR2A
SCHEMBL24858602 0.79 DAO (0.44) GABRA1GABRB2DAOELANEFLT3
SCHEMBL26708797 0.78 GABRA1 (0.42) GABRA1GABRB2DAOELANEFLT3
SCHEMBL5748520 0.77 ELANE (0.46) GABRA1GABRB2DAOELANEKDM4E
SCHEMBL24697255 0.77 GABRA1 (0.41) GABRA1GABRB2DAOFLT3ESR1
SCHEMBL25079343 0.77 GABRA1 (0.41) GABRA1GABRB2DAOELANEFLT3
SCHEMBL24680252 0.77 GABRA1 (0.41) GABRA1GABRB2DAOELANEFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192790-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2022-09-15 WO disclosed