SCHEMBL24697998

SCHEMBL24697998

Oc1nc(Cl)nc2c1CCC2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.40
MAPK1 P28482 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
BPTF Q12830 1/20 0.40
NSD2 O96028 1/20 0.36
GRIN1 Q05586 7/20 0.35
GRIN2A Q12879 7/20 0.35
BCHE P06276 6/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
CASP6 P55212 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574606 0.96 ACHE (0.41) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL633261 0.77 ACHE (0.43) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL30777931 0.77 ACHE (0.43) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL30350953 0.77 ACHE (0.43) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL1821069 0.77 ACHE (0.43) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL13394086 0.74 KDM4E (0.53) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL1586850 0.74 KDM4E (0.53) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL18711586 0.74 KDM4E (0.41) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL191381 0.74 ACHE (0.40) ACHEMAPK1MEN1KMT2ABPTF
SCHEMBL9267023 0.74 ACHE (0.50) ACHEMAPK1MEN1KMT2ABPTF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed