SCHEMBL24698018

SCHEMBL24698018

C[C@H]1CCN1c1nc2c(c(-c3cccnc3)n1)CCC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
PIK3CA P42336 1/20 0.39
KDM4E B2RXH2 2/20 0.38
HTT P42858 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
MTOR P42345 1/20 0.37
ALDH1A1 P00352 2/20 0.37
TP53 P04637 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
CDK19 Q9BWU1 1/20 0.37
MAPK1 P28482 1/20 0.36
USP1 O94782 1/20 0.36
WDR48 Q8TAF3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015307 1.00 HRH3 (0.48) HRH3PIK3CAKDM4EHTTHSD17B10
SCHEMBL24698056 0.87 PIK3CA (0.35) HRH3PIK3CAKDM4EMEN1KMT2A
SCHEMBL24698168 0.87 HRH2 (0.43) HRH3KDM4EHSD17B10MEN1KMT2A
SCHEMBL24698853 0.85 ALDH1A1 (0.37) HRH3PIK3CAKDM4EHSD17B10TSHR
SCHEMBL24697693 0.85 MEN1 (0.34) HRH3PIK3CAKDM4EMEN1KMT2A
SCHEMBL30016322 0.82 BRD4 (0.36) HRH3PIK3CAMEN1KMT2AMTOR
SCHEMBL24697563 0.82 BRD4 (0.36) HRH3PIK3CAMEN1KMT2AMTOR
SCHEMBL24699331 0.82 MEN1 (0.39) HRH3KDM4EHSD17B10MEN1KMT2A
SCHEMBL30015772 0.82 MEN1 (0.39) HRH3KDM4EHSD17B10MEN1KMT2A
SCHEMBL24698400 0.82 PIK3CA (0.49) HRH3PIK3CAKDM4EHTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed