SCHEMBL24698181

SCHEMBL24698181

CC(C)(O)c1ccc(-c2nc(N3CC(O)C3)nc3c2CCC3)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 3/20 0.38
PDE10A Q9Y233 1/20 0.38
WNT3A P56704 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
HRH2 P25021 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TNF P01375 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
KDM4E B2RXH2 4/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
PDK1 Q15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698835 0.87 GBA1 (0.47) GBA1WNT3ATNKS2HRH2HRH3
SCHEMBL24698179 0.84 WNT3A (0.36) GBA1PDE10AWNT3ATNKS2HRH2
SCHEMBL24698834 0.81 WNT3A (0.36) GBA1WNT3ATNKS2HRH2HRH3
SCHEMBL24698426 0.80 KARS1 (0.40) GBA1HRH2HRH3KDM4EALDH1A1
SCHEMBL24698113 0.80 HRH2 (0.36) HRH2HRH3KDM4EMAPTLMNA
SCHEMBL24699432 0.80 HRH2 (0.38) HRH2HRH3KDM4EMAPTLMNA
SCHEMBL24698868 0.79 PDE2A (0.38) GBA1PDE10AHRH2HRH3KDM4E
SCHEMBL24697726 0.77 HRH2 (0.34) HRH2HRH3KDM4EMAPTLMNA
SCHEMBL24699404 0.76 NISCH (0.35) HRH2HRH3KDM4EMAPTLMNA
SCHEMBL24697711 0.76 KHK (0.43) HRH2HRH3KDM4EMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed