SCHEMBL24698802

SCHEMBL24698802

C[C@H]1CCN1c1nc2c(c(-c3ccnc(F)c3)n1)CCC2

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.40
MAP3K12 Q12852 6/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
TRPV1 Q8NER1 2/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
KCNH2 Q12809 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
GRM2 Q14416 1/20 0.32
PARP10 Q53GL7 1/20 0.32
PARP11 Q9NR21 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016131 1.00 MTOR (0.40) MTORMAP3K12KDM4EMAPTTRPV1
SCHEMBL24698853 0.84 ALDH1A1 (0.37) MTORKDM4EMAPTTRPV1HRH3
SCHEMBL24698177 0.84 PDE4A (0.35) MTORMAP3K12GRM2
SCHEMBL29134519 0.83 PIK3R1 (0.35) MAP3K12PDK1PDK2PDK3PDK4
SCHEMBL30016476 0.83 PIK3R1 (0.35) MAP3K12PDK1PDK2PDK3PDK4
SCHEMBL24697783 0.83 PIK3R1 (0.35) MAP3K12PDK1PDK2PDK3PDK4
SCHEMBL24698813 0.82 IGF1R (0.37) KDM4EMAPTPARP10PARP11
SCHEMBL30015981 0.81 TGFBR1 (0.40) MAP3K12
SCHEMBL24697693 0.81 MEN1 (0.34) MAP3K12KDM4ETRPV1PDK1PDK2
SCHEMBL30015933 0.81 MAP4K4 (0.37) MAP3K12KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed