SCHEMBL24699059

SCHEMBL24699059

COc1ccc(-c2nc(N3CC[C@@H]3C)nc3c2CCC3)cc1S(=N)(=O)c1ccc(C#N)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.34
HSD17B10 Q99714 3/20 0.34
USP2 O75604 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HPGD P15428 1/20 0.33
MTOR P42345 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
PDE5A O76074 8/20 0.33
BRD4 O60885 2/20 0.33
BRD1 O95696 2/20 0.33
BRPF1 P55201 2/20 0.33
BRD9 Q9H8M2 2/20 0.33
BRPF3 Q9ULD4 2/20 0.33
PDE6D O43924 1/20 0.32
PDE6A P16499 1/20 0.32
PDE6G P18545 1/20 0.32
PDE6B P35913 1/20 0.32
PDE6C P51160 1/20 0.32
PDE6H Q13956 1/20 0.32
ALPL P05186 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30014813 1.00 MAPK1 (0.34) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699069 0.93 PI4KB (0.35) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30015941 0.93 PI4KB (0.35) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30016531 0.89 PI4KB (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24697976 0.89 PI4KB (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699210 0.87 MTOR (0.35) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30015825 0.87 MTOR (0.35) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699229 0.84 MTOR (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30016058 0.84 MTOR (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699239 0.82 HMOX1 (0.34) MTORBRD4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed