SCHEMBL24699358

SCHEMBL24699358

NC(=O)c1ccc(Br)cc1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.49
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
PLA2G2A P14555 4/20 0.46
PLA2G10 O15496 3/20 0.46
ADRA1D P25100 1/20 0.46
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
RXFP1 Q9HBX9 1/20 0.43
PTPN1 P18031 3/20 0.43
PARP15 Q460N3 2/20 0.43
PARP10 Q53GL7 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN6 P29350 1/20 0.43
SLCO1B1 Q9Y6L6 1/20 0.42
BCL2 P10415 1/20 0.42
BCL2L1 Q07817 1/20 0.42
CDC7 O00311 1/20 0.42
MPO P05164 1/20 0.41
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015569 1.00 DGAT1 (0.49) DGAT1HPGDKMT2APLA2G2APLA2G10
SCHEMBL27757808 0.87 HPGD (0.49) HPGDKMT2APOLBMAPTPTPN1
SCHEMBL3303005 0.87 PTPN1 (0.53) HPGDKMT2APOLBMAPTRXFP1
SCHEMBL10827633 0.84 KMT2A (0.47) HPGDKMT2APLA2G2APLA2G10POLB
SCHEMBL6140508 0.82 PLA2G2A (0.61) PLA2G2APLA2G10POLBMAPTPTPN1
SCHEMBL3053719 0.81 BCL2 (0.40) HPGDKMT2AADRA1DPOLBMAPT
SCHEMBL3091338 0.81 PARP15 (0.48) DGAT1HPGDKMT2APOLBMAPT
SCHEMBL2428547 0.81 PLA2G2A (0.57) PLA2G2APLA2G10PTPN1PTPN2PTPN6
SCHEMBL5802389 0.81 PLA2G2A (0.46) PLA2G2APLA2G10PTPN1PARP10PTPN2
SCHEMBL28838076 0.81 MEN1 (0.58) HPGDKMT2APLA2G2APLA2G10ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260092053-A1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2026-04-02 US disclosed
EP-4681774-A2 KHK INHIBITORS Gilead Sciences, Inc. (US) 2026-01-21 EP disclosed
EP-4313967-B1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2025-11-12 EP disclosed
US-12410160-B2 KHK inhibitors GILEAD SCIENCES, INC. (US) 2025-09-09 US disclosed
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
US-20230079863-A1 KHK INHIBITORS GILEAD SCIENCES, INC. 2023-03-16 US disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260092053-A1 KHK INHIBITORS KHK, SLC5A2, HK1 DGAT1 1085/4885HPGD 3162/4885KMT2A 1037/4885
US-20230079863-A1 KHK INHIBITORS KHK, KHDRBS1, NADK DGAT1 3451/4885HPGD 1949/4885KMT2A 283/4885
US-12410160-B2 KHK inhibitors KHK, KHDRBS1, NADK DGAT1 3451/4885HPGD 1949/4885KMT2A 283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.