SCHEMBL6140508

SCHEMBL6140508

NC(=O)c1ccc(C(N)=O)c(Cc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 4/20 0.61
PLA2G10 O15496 3/20 0.61
BCL2 P10415 1/20 0.47
BCL2L1 Q07817 1/20 0.47
TSHR P16473 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
MBTD1 Q05BQ5 1/20 0.45
L3MBTL3 Q96JM7 1/20 0.45
PARP10 Q53GL7 1/20 0.45
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
JAK3 P52333 1/20 0.44
PTPN1 P18031 2/20 0.44
PTPN2 P17706 1/20 0.44
PTPN6 P29350 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
PARP1 P09874 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2428547 0.92 PLA2G2A (0.57) PLA2G2APLA2G10BCL2BCL2L1TSHR
SCHEMBL16584765 0.92 PLA2G2A (0.59) PLA2G2APLA2G10BCL2BCL2L1TSHR
SCHEMBL6141261 0.87 PARP10 (0.58) PLA2G2APLA2G10PARP10
SCHEMBL8581956 0.86 PLA2G10 (0.42) PLA2G2APLA2G10TSHRL3MBTL1PARP10
SCHEMBL28309719 0.84 CYP17A1 (0.58) PLA2G2APLA2G10JAK2JAK1TYK2
SCHEMBL28309715 0.82 F7 (0.49) CYP3A4MAPTRECQL
SCHEMBL24699358 0.82 DGAT1 (0.49) PLA2G2APLA2G10BCL2BCL2L1PARP10
SCHEMBL5802389 0.82 PLA2G2A (0.46) PLA2G2APLA2G10BCL2BCL2L1PARP10
SCHEMBL14720212 0.82 PLA2G2A (0.59) PLA2G2APLA2G10BCL2BCL2L1TSHR
SCHEMBL28838076 0.82 MEN1 (0.58) PLA2G2APLA2G10BCL2BCL2L1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1497260-A1 NOVEL METHOXYBENZAMIDE COMPOUNDS FOR USE IN MCH RECEPTOR RELATED DISORDERS 7TM Pharma A/S (DK) 2005-01-19 EP disclosed
WO-2004048319-A1 NOVEL BENZAMIDE COMPOUNDS FOR USE IN MCH RECEPTOR RELATED DISORDERS 7TM PHARMA A/S (DK) 2004-06-10 WO disclosed
WO-2003087045-A1 NOVEL METHOXYBENZAMIDE COMPOUNDS FOR USE IN MCH RECEPTOR RELATED DISORDERS 7TM PHARMA A/S (DK) 2003-10-23 WO disclosed