SCHEMBL24699490

SCHEMBL24699490

c1cc(-c2nc(N3CCC3)nc3c2CCC3)ncn1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GSK3B P49841 1/20 0.38
PIK3CA P42336 1/20 0.36
IGF1R P08069 6/20 0.36
GBA1 P04062 2/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
CDC42BPB Q9Y5S2 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698701 0.83 TDP1 (0.41) KDM4EALDH1A1GBA1SMN1; SMN2LMNA
SCHEMBL24699489 0.82 GSK3B (0.35) ALDH1A1GSK3BLMNA
SCHEMBL30015011 0.82 GSK3B (0.35) ALDH1A1GSK3BLMNA
SCHEMBL24698856 0.81 PIK3CA (0.47) KDM4EALDH1A1PIK3CAIGF1RGBA1
SCHEMBL24699070 0.80 ALDH1A1 (0.39) KDM4EALDH1A1IGF1RGBA1HPGD
SCHEMBL19623360 0.77 PIK3CA (0.46) KDM4EALDH1A1PIK3CAIGF1RGBA1
SCHEMBL24698057 0.75 PIK3CA (0.44) KDM4EALDH1A1PIK3CAIGF1RGBA1
SCHEMBL24697574 0.75 KDM4E (0.39) KDM4EALDH1A1IGF1RGBA1HPGD
SCHEMBL24698050 0.75 IGF1R (0.41) KDM4EALDH1A1IGF1RGBA1HPGD
SCHEMBL24699355 0.75 KDM4E (0.42) KDM4EALDH1A1PIK3CAIGF1RGBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed