SCHEMBL24699495

SCHEMBL24699495

COc1cc(-c2nc(N3CC[C@@H]3C)nc3c2CCC3)ccc1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.41
HSD17B10 Q99714 3/20 0.41
USP2 O75604 1/20 0.41
KDM4E B2RXH2 4/20 0.40
HPGD P15428 1/20 0.40
MTOR P42345 1/20 0.40
LMNA P02545 1/20 0.39
S1PR1 P21453 1/20 0.38
AR P10275 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
PGR P06401 2/20 0.36
NR3C2 P08235 1/20 0.36
NSD2 O96028 1/20 0.36
HRH2 P25021 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KDM1A O60341 2/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015914 1.00 MAPK1 (0.41) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699229 0.86 MTOR (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30016058 0.86 MTOR (0.36) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL30016865 0.86 AR (0.36) KDM4EHPGDARALDH1A1GAA
SCHEMBL24698160 0.86 AR (0.36) KDM4EHPGDARALDH1A1GAA
SCHEMBL30016357 0.86 MTOR (0.44) MTORKDM1A
SCHEMBL24699037 0.86 MTOR (0.44) MTORKDM1A
SCHEMBL24699497 0.85 HSD17B10 (0.43) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699243 0.85 KDM1A (0.33) MAPK1HSD17B10USP2KDM4EHPGD
SCHEMBL24699484 0.82 PDE7A (0.41) MAPK1HSD17B10USP2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed