SCHEMBL30016865

SCHEMBL30016865

C[C@H]1CCN1c1nc2c(c(-c3ccc(C#N)c(Cl)c3)n1)CCC2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.36
CYP11B2 P19099 3/20 0.36
NR3C2 P08235 3/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
NSD2 O96028 1/20 0.34
KDM1A O60341 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
GAA P10253 1/20 0.33
EGLN2 Q96KS0 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698160 1.00 AR (0.36) ARCYP11B2NR3C2PDK1PDK2
SCHEMBL24699037 0.88 MTOR (0.44) CYP11B2KDM1A
SCHEMBL30016357 0.88 MTOR (0.44) CYP11B2KDM1A
SCHEMBL30015914 0.86 MAPK1 (0.41) ARNR3C2KDM4EALDH1A1HPGD
SCHEMBL24699495 0.86 MAPK1 (0.41) ARNR3C2KDM4EALDH1A1HPGD
SCHEMBL24698161 0.84 CYP11B2 (0.39) ARCYP11B2KDM4EALDH1A1HPGD
SCHEMBL30015825 0.82 MTOR (0.35) NR3C2KDM4EHPGDKDM1A
SCHEMBL24698381 0.82 MTOR (0.41) ALDH1A1HPGDHRH3
SCHEMBL29134822 0.82 MTOR (0.41) ALDH1A1HPGDHRH3
SCHEMBL30014710 0.82 MTOR (0.41) ALDH1A1HPGDHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed