SCHEMBL24715944

SCHEMBL24715944

COc1ccc(F)c2ccoc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
HPGD P15428 5/20 0.50
LMNA P02545 4/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
KDM4E B2RXH2 6/20 0.44
CYP3A4 P08684 5/20 0.44
HSD17B10 Q99714 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 3/20 0.38
TP53 P04637 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 1/20 0.37
KCNA3 P22001 4/20 0.37
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 2/20 0.37
POLB P06746 1/20 0.37
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12804046 0.85 ALDH1A1 (0.42) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL28125752 0.84 ALDH1A1 (0.56) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL8358409 0.78 ALDH1A1 (0.51) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL789045 0.77 ALDH1A1 (0.50) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL1747096 0.77 ALDH1A1 (0.50) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL28731604 0.74 ALOX15 (0.42) ALDH1A1HPGDLMNAKMT2AKDM4E
SCHEMBL2992833 0.73 ALDH1A1 (0.50) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL2122119 0.73 IMPDH2 (0.54) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL3253868 0.72 ALDH1A1 (0.49) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL806499 0.71 ALDH1A1 (0.43) ALDH1A1HPGDLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761410-B Pyrrolopyrimidinone compounds and application thereof 广州必贝特医药股份有限公司 2023-08-25 CN disclosed
WO-2022213932-A1 PYRROLOPYRIMIDINONE COMPOUND AND APPLICATION THEREOF 广州必贝特医药股份有限公司 2022-10-13 WO disclosed
WO-2022179469-A1 THIENOPYRIMIDINEDIONE COMPOUNDS AND APPLICATION THEREOF 南京明德新药研发有限公司 2022-09-01 WO disclosed
CN-114761410-A Pyrrolopyrimidinone compounds and application thereof 广州必贝特医药股份有限公司 2022-07-15 CN disclosed